|  | n | Dose | Dose/body weight | C0 | Cmax | AUC0-12 | AUC0-12 / Dose | AUC0-0.5 |
---|---|---|---|---|---|---|---|---|---|
(mg) | (mg/kg) | (μg/mL) | (μg/mL) | (μg∙h/mL) | (μg∙h/mL/mg) | (μg∙h/mL) | |||
Gastrointestinal involvement |  +  | 10 | 1500 (1500–1500) | 28.3 (25.8–30.9) | 1.9 (1.3–3.1) | 26.3* (15.4–29.7) | 63.4* (53.8–89.4) | 0.049 (0.031–0.062) | 6.3** (4.2–7.9) |
 −  | 23 | 1500 (1500–1875) | 227.6 (23.6–35.0) | 1.8 (1.2–2.8) | 12.3 (8.7–19.7) | 45.3 (34.8–68.4) | 0.030 (0.024–0.052) | 2.9 (1.0–3.7) | |
Infection |  +  | 14 | 1500 (1500–1875) | 28.5 (26.3–33.2) | 1.6 (1.2–3.2) | 17.0 (10.9–23.5) | 49.7 (41.3–77.8) | 0.028 (0.024–0.047) | 3.3 (2.5–3.9) |
 −  | 19 | 1500 (1500–1625) | 27.3 (21.9–34.6) | 1.9 (1.2–2.6) | 12.8 (10.4–27.7) | 51.1 (40.8–68.4) | 0.036 (0.030–0.061) | 3.7 (1.1–6.6) |